Tom ntej: Retatrutide Peptide CAS 2381089-83-2

Tom ntej: Retatrutide Peptide CAS 2381089-83-2
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Khoom npe: Retatrutide Peptide Powder
CAS Nr .: 2592008-21-0
Cov tsos mob: Dawb, tsis muaj menyuam, lyophilized hmoov
Cov mis mos molecular: C215H347N61O65
Molecular Luj: 4,852.5
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Tom ntej: Retatrutide Peptide CAS 2381089-83-2

 

Khoom npe Retatrutide Peptide Hmoov
CAS Nr 2592008-21-0
Qhov tshwm sim Dawb, sterile, lyophilized hmoov
Molecular Formula C215H347N61O65
Molecular Luj 4,852.50
Purity (HPLC) Ntau dua lossis sib npaug li 99% (Tsev Tshuaj)
Txee lub neej 24 lub hlis ( khaws cia ntawm -20 degree, tiv thaiv los ntawm lub teeb)
Kev kho dua tshiab PBS tsis kam (pH 7.4)
Ntim Lub raj mis kaw
Yam tsawg kawg nkaus Order Quantity 1 g (ntau ntau muaj)

 

Retatrutide Peptide 99%:Triple -Agonist Revolutionizing Metabolic Disease Treatment
-Global First GLP-1R/GIPR/GCGR Triple Agonist for Obesity, Diabetes, thiab NASH

 

Retatrutide Peptide Specifications

 

Retatrutide peptide hmoov yog ib qho hluavtaws 39-amino acid peptide engineered rau stability, multi-receptor affinity, thiab ncua ib nrab-lub neej. Nws cov qauv sib txuas cov ntsiab lus los ntawm GLP-1, GIP, thiab glucagon (GCG) los tsim ib qho triple agonist nrog optimized pharmacokinetics.
Retatrutide peptide sawv cev rau kev hloov pauv hloov pauv los ntawm kev sib koom ua ke ntawm peb qhov tseem ceeb receptors koom nrog hauv kev tswj cov piam thaj, tswj kev qab los noj mov, thiab kev siv hluav taws xob.

 

Yuav Ua Li Cas Retatrutide Peptide Ua Haujlwm

Retatrutide Peptide's triple agonism tsim ib qho kev sib koom ua ke uas hais txog kev rog rog, hyperglycemia, thiab daim siab rog ntau ntxiv:

GLP-1 Receptor Activation

  • Stimulates insulin secretion los ntawm pancreatic -cov cell hauv cov piam thaj- nyob ntawm seb.
  • inhibits glucagon tso tawm los ntawm -cells, txo cov piam thaj hauv siab.
  • Ua kom lub plab zom mov qeeb, txhim kho satiety thiab txo cov khoom noj.

GIP Receptor Activation

  • Txhim kho cov ntaub so ntswg adipose lipolysis, tso cov fatty acids dawb rau kev siv lub zog.
  • Txhim kho insulin rhiab heev hauv cov leeg pob txha thiab daim siab, tiv thaiv insulin tsis kam.
  • Txo cov hepatic triglyceride synthesis, txo cov roj siab hauv siab.

Ua kom GCGR

  • Ua kom cov thermogenesis ntawm xim av adipose cov ntaub so ntswg, txhawb kev siv calorie.
  • Txhawb glycogenolysis thiab lipolysis, txhawb nqa lub zog.
  • Txo cov hepatic steatosis los ntawm inhibiting de novo lipogenesis.

Clinical Advantage: Thaum Semaglutide thiab Tirzepatide modulate 1-2 txoj hauv kev, Retatrutide Peptide's triple agonism ua tiav kev poob phaus, tswj glycemic, thiab daim siab rog txo los ntawm kev hais txog tag nrho peb lub ntsiab lus ntawm metabolic tsis ua haujlwm ib txhij.

 

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Cov ntaub ntawv kho mob dab tsi qhia txog Retatrutide peptide

Poob Poob ntawm Retatrutide peptide Powder: Teem Cov Qauv Tshiab

Theem II Trial (N=338, 48 lub lis piam):

  • 12 mg koob: 24.2% qhov hnyav poob qis (vs . 22.5% rau Tirzepatide thiab 16% rau Semaglutide).
  • Ntau dua lossis sib npaug li 20% poob phaus: 63% ntawm cov neeg mob (vs . 50% rau Tirzepatide thiab 34% rau Semaglutide).
  • Ntau dua lossis sib npaug li 30% poob phaus: 25% ntawm cov neeg mob (tsis tau pom dua hauv kev sim tshuaj tshuaj).
 

Glycemic Control ntawm Retatrutide peptide Powder: HbA1c Txo

Phase II sim (T2D Cov Neeg Mob, 36 lub lis piam):

  • 12 mg koob: 2.5–3.0% txo HbA1c (vs. 1.5–2.0% rau Semaglutide thiab Tirzepatide).
  • Kev Kho Mob Ntshav Qab Zib: 40% ntawm cov neeg mob ua tiav HbA1c<6.5% without medication.
 

Kev txo qis hauv siab ntawm Retatrutide peptide Powder: NASH Kev Kho Mob Muaj Peev Xwm

Theem II Kev sim (NAFLD Cov Neeg Mob, 24 lub lis piam):

  • Cov ntsiab lus rog hauv siab: 86% txo (MRI- ntsuas PDFF) vs . 50–60% rau Semaglutide/Tirzepatide.
  • ALT / AST theem: normalized nyob rau hauv 70% ntawm cov neeg mob, qhia tias txo daim siab mob.
 

 

Retatrutide peptide VS Tirzepatide VS Semaglutide

 

product-1143-281

 

Kev sib piv

Semaglutide

Tirzepatide

Retatrutide

Mechanism ntawm Action

Tib - lub hom phiaj: Ua rau GLP-1 receptor

Dual -target: Ua kom GLP-1 + GIP receptors

Triple -target: Ua kom GLP-1 + GIP + GCGR receptors

Core Functions

Txhawb nqa insulin secretion, inhibits glucagon, qeeb plab hnyuv

Txhim kho insulin secretion, txhim kho insulin rhiab heev, txo cov kev mob tshwm sim GI

Boosts metabolism (fat so + zog siv), ncaj qha hlawv rog, txo daim siab rog

Poob Qhov Ua Tau Zoo

15% -18% txo qhov nruab nrab (68 lub lis piam)

18% -22.5% txo qhov nruab nrab (72 lub lis piam)

24.2% txo qhov nruab nrab (48 lub lis piam; 63% ua tiav Ntau dua lossis sib npaug li 20% poob phaus)

Kev txhim kho metabolic

Txo HbA1c, txhim kho glycemic tswj

Txo HbA1c, txo lub siab rog (zoo dua rau Semaglutide)

86% daim siab txo qis (24 lub lis piam); 40% txo qis ntshav qab zib

Kev ua lag luam Positioning

Thawj -cov tshuaj poob phaus rau pob nyiaj- cov neeg mob tsis nco qab

Hwm dual - lub hom phiaj kev xaiv rau cov neeg mob metabolic syndrome

Qhov kawg poob phaus + metabolic breakthrough, yav tom ntej ua lag luam thawj coj

 

Cov Lus Cim Tseem Ceeb:

Mechanism ntawm Action

Retatrutide Peptide's triple - lub hom phiaj tsim (GLP-1/GIP/GCGR) yog nws qhov zoo tshaj plaws, nrog GCGR ua kom ncaj qha txhawb kev rog rog.

Poob Qhov Ua Tau Zoo

Retatrutide Peptide cov ntaub ntawv 48-lub lim tiam ua tau zoo tshaj 72-lub lim tiam cov txiaj ntsig ntawm nws cov neeg sib tw, qhia tau sai thiab muaj zog dua.

Kev txhim kho metabolic

Retatrutide Peptide Powderexcels hauv daim siab txo qis thiab txo cov ntshav qab zib, ua rau nws zoo tagnrho rau cov neeg mob NASH thiab metabolic syndrome.

product-1100-733

 

Vim li cas thiaj xaiv Peb Retatrutide peptide Hmoov?

01/

Quality Assurance:
Purity Ntau dua lossis sib npaug li 99%, endotoxin<0.1 EU/mg, and stability data (2-year shelf life at -20°C).

02/

Txoj Cai Ua Raws Cai:
Thov COA, MSDS, DSC (cov ntaub ntawv qhia txog kev ruaj ntseg), thiab kev kuaj mob IDs (xws li, NCT tooj).

03/

Logistics:
Peb cov kev pabcuam logistics lav kev nyab xeeb, kev xa khoom sai thoob ntiaj teb, thaum muab kev lis kev cai dual (DDP) nrog rau tag nrho cov se them ua ntej thiab qhov rooj-rau- qhov rooj yooj yim.

04/

Customizable Formulations:
Cov tshuaj kho kom haum (1 mg–1 kg) rau R&D lossis siv coj mus muag.

 

Tiv tauj peb
Retatrutide peptide Powder redefines thaj chaw kho mob rau kev rog rog, ntshav qab zib, thiab NASH los ntawm kev sib koom ua ke GLP-1R, GIPR, thiab GCGR agonism rau hauv ib qho molecule. Nws qhov kev poob phaus tsis tau pom dua (24.2%), kev tswj hwm glycemic zoo dua, thiab txo qis hauv siab ua rau nws ua tus thawj coj hauv kev lag luam tshuaj metabolic $ 100 billion.
Rau cov lus nug ntau lossis cov qauv kev cai, hu rau peb pab neeg niaj hnub no kom ruaj ntseg koj cov khoom siv ntawm cov khoom siv tshuaj hloov pauv no.

 

Cim npe nrov: Tuam Tshoj Retatrutide Peptide CAS 2381089-83-2 Chaw tsim tshuaj paus, lwm tus neeg, Hoobkas

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